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\psz9\linex0\headery709\footery709\colsx284\endnhere\sectdefaultcl\sectrsid12468991\sftnbj {\rtlch\fcs1 \af1\afs24 \ltrch\fcs0 \fs24\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid9721414
\par }\pard \ltrpar\qj \li0\ri-1\sl360\slmult1\widctlpar\wrapdefault\faauto\adjustright\rin-1\lin0\itap0\pararsid12468991 {\rtlch\fcs1 \af1\afs24 \ltrch\fcs0 \fs24\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid9721414 NPD1 was shown to }{\rtlch\fcs1
\ab\af1\afs24 \ltrch\fcs0 \fs24\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid9721414 participate to the active process of resolution of inflammation}{\rtlch\fcs1 \af1\afs24 \ltrch\fcs0
\fs24\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid9721414 . It reduces neutrophil accumulation and infiltration, and it is}{\rtlch\fcs1 \ab\af1\afs24 \ltrch\fcs0 \fs24\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid9721414
implicated in the return to cellular homeostasis,}{\rtlch\fcs1 \af1\afs24 \ltrch\fcs0 \fs24\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid9721414 included wound healing.
\par Since}{\rtlch\fcs1 \ab\af1\afs24 \ltrch\fcs0 \fs24\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid9721414 inflammation}{\rtlch\fcs1 \af1\afs24 \ltrch\fcs0 \fs24\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid9721414
is a very complex multi-factorial process which plays a crucial role in many major current diseases such as }{\rtlch\fcs1 \ab\af1\afs24 \ltrch\fcs0 \fs24\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid9721414 Alzheimer\rquote s}{\rtlch\fcs1
\af1\afs24 \ltrch\fcs0 \fs24\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid9721414 disease, }{\rtlch\fcs1 \ab\af1\afs24 \ltrch\fcs0 \fs24\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid9721414 atherosclerosis}{\rtlch\fcs1 \af1\afs24
\ltrch\fcs0 \fs24\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid9721414 , }{\rtlch\fcs1 \ab\af1\afs24 \ltrch\fcs0 \fs24\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid9721414 cancers}{\rtlch\fcs1 \af1\afs24 \ltrch\fcs0
\fs24\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid9721414 , }{\rtlch\fcs1 \ab\af1\afs24 \ltrch\fcs0 \fs24\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid9721414 cardiovascular}{\rtlch\fcs1 \af1\afs24 \ltrch\fcs0
\fs24\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid9721414 diseases, chronic }{\rtlch\fcs1 \ab\af1\afs24 \ltrch\fcs0 \fs24\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid9721414 asthma}{\rtlch\fcs1 \af1\afs24 \ltrch\fcs0
\fs24\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid9721414 , }{\rtlch\fcs1 \ab\af1\afs24 \ltrch\fcs0 \fs24\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid9721414 arthritis}{\rtlch\fcs1 \af1\afs24 \ltrch\fcs0
\fs24\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid9721414 , etc., further investigation of this polyunsaturated metabolite }{\rtlch\fcs1 \af1\afs24 \ltrch\fcs0 \fs24\lang2057\langfe1031\langnp2057\insrsid8345954 and its analogs are}{\rtlch\fcs1
\af1\afs24 \ltrch\fcs0 \fs24\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid9721414 of great interest.
\par }{\rtlch\fcs1 \ab\af1\afs24 \ltrch\fcs0 \fs24\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid9721414 However, }{\rtlch\fcs1 \af1\afs24 \ltrch\fcs0 \fs24\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid9721414
for lack of standards in sufficient quantities, detection and quantification of this new endogenous lipid mediator in enflamed tissues, but also studies on the mechanism of its action (receptors, location, etc.) cannot be performed }{\rtlch\fcs1
\ab\af1\afs24 \ltrch\fcs0 \fs24\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid9721414 efficiently}{\rtlch\fcs1 \af1\afs24 \ltrch\fcs0 \fs24\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid9721414 . Effectively, it is }{\rtlch\fcs1
\ab\af1\afs24 \ltrch\fcs0 \fs24\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid9721414 not commercially available}{\rtlch\fcs1 \af1\afs24 \ltrch\fcs0 \fs24\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid9721414
and extractions of biological tissues provide tiny amounts only, thus restricting the number and the types of biological experiments. Furthermore, it is noteworthy that the }{\rtlch\fcs1 \af1\afs24 \ltrch\fcs0
\fs24\lang2057\langfe1031\langnp2057\insrsid9721414 in vitro}{\rtlch\fcs1 \af1\afs24 \ltrch\fcs0 \fs24\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid9721414 enzymatic synthesis (}{\rtlch\fcs1 \af1\afs24 \ltrch\fcs0
\fs24\lang2057\langfe1031\langnp2057\insrsid9721414 in vitro}{\rtlch\fcs1 \af1\afs24 \ltrch\fcs0 \fs24\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid9721414 ) starting from }{\rtlch\fcs1 \af1\afs24 \ltrch\fcs0
\fs24\lang2057\langfe1031\langnp2057\insrsid11479346 DHA}{\rtlch\fcs1 \af1\afs24 \ltrch\fcs0 \fs24\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid9721414 and lipoxygenases did not yield to the expected NPD1 but to an isomer (called PDX) }{
\rtlch\fcs1 \af1\afs24 \ltrch\fcs0 \fs24\lang2057\langfe1031\langnp2057\insrsid9721414 showing a E,Z,}{\rtlch\fcs1 \af1\afs24 \ltrch\fcs0 \fs24\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid9721414
E-triene unit instead of the desired Z,E,E-triene unit.}{\field\fldedit{\*\fldinst {\rtlch\fcs1 \af1\afs24 \ltrch\fcs0 \fs24\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid9721414
ADDIN EN.CITE Chen200988<
REFERENCE_TYPE>088Chen, P.Fenet, B.Michaud, S.Tomczyk, N.Vericel, E.Lagarde, M.Guichardant, M.
2009Full characterization of PDX, a neuroprotectin/protectin D1 isomer, which inhibits blood platelet aggregationFEBS Lett583213478-3484-NPD2009lo4Nov 319818771triene EZE protectin - voir la thèse Villeurbanne correspondanteArachidonate 15-Lipoxygenase/metabolismCarbon/chemistryDocosahexaenoic Acids/*chemistry/metabolism/*pharmacologyDose-Response Relationship, DrugGas Chromatography-Mass Spectro
m
etryHumansHydroxides/chemistryMagnetic Resonance SpectroscopyPlatelet Aggregation/*drug effectsSoybeans/enzymologyStereoisomerism
K
EYWORDS>http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&dopt=Citation&list_uids=19818771Universite de Lyon, Inserm UMR 870, Insa-Lyon, RMND/IMBL, Inra 1235, 69621 Villeurbanne, France.Butovich2006-NPD2006lo636036Butovich, I. A.
s
tyles>2006-NPD2006lo6A one-step method of 10,17-dihydro(pero)xydocosahexa-4Z,7Z,11E,13Z,15E,19Z-enoic acid synthesis by soybean lipoxygenaseJ Lipid Res474854
-
863Apr16391324Chromatography, High Pressure LiquidDocosahexaenoic Acids/chemistry/*metabolismLipoxygenase/*metaboli
s
mMolecular StructureOxidation-ReductionPlant Proteins/metabolismSoybeans/*enzymologyhttp://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=Pub
Med&dopt=Citation&list_uids=16391324Department of Ophthalmology, University of Texas Southwestern Medical Center, Dallas, TX 75390-9057, USA. igor.butovich@utsouthwestern.edu}
}{\fldrslt {\rtlch\fcs1 \af1\afs24 \ltrch\fcs0 \fs24\lang2057\langfe1031\super\langnp2057\insrsid9721414\charrsid9721414 2,3}}}\sectd \ltrsect\psz9\linex0\headery709\footery709\colsx284\endnhere\sectdefaultcl\sectrsid12468991\sftnbj {\rtlch\fcs1
\af1\afs24 \ltrch\fcs0 \fs24\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid9721414
\par }\pard \ltrpar\qj \li0\ri-1\sl360\slmult1\widctlpar\wrapdefault\faauto\rin-1\lin0\itap0\pararsid12468991 {\rtlch\fcs1 \ab\af1\afs24 \ltrch\fcs0 \fs24\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid9721414 Thus,
we performed a total synthesis of a NPD1 epimer using a flexible strategy that can give access to different diastereoisomers, isomers or analogs.
\par }\pard \ltrpar\qj \li0\ri-1\sl360\slmult1\widctlpar\wrapdefault\faauto\adjustright\rin-1\lin0\itap0\pararsid12468991 {\rtlch\fcs1 \af1\afs24 \ltrch\fcs0 \fs24\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid9721414
The proposed strategy features Wittig olefinations, }{\rtlch\fcs1 \af1\afs24 \ltrch\fcs0 \fs24\lang2057\langfe1031\langnp2057\insrsid8549655 Colvin rearrangement, hydrometalation}{\rtlch\fcs1 \af1\afs24 \ltrch\fcs0
\fs24\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid9721414 , Sonogashira cross coupling reactions.
\par }{\rtlch\fcs1 \ab\af1\afs16 \ltrch\fcs0 \b\fs16\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid2766518
\par }{\rtlch\fcs1 \ab\af1\afs20 \ltrch\fcs0 \b\fs20\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid12468991 References
\par }\pard \ltrpar\qj \fi-142\li142\ri0\widctlpar\wrapdefault\faauto\adjustright\rin0\lin142\itap0\pararsid12468991 {\field\fldedit{\*\fldinst {\rtlch\fcs1 \ab\af1\afs20 \ltrch\fcs0 \fs20\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid12468991
ADDIN EN.REFLIST }}{\fldrslt {\rtlch\fcs1 \ab\af1\afs20 \ltrch\fcs0 \fs20\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid12468991 (1) }{\rtlch\fcs1 \ab\af1\afs20 \ltrch\fcs0 \fs20\lang2057\langfe1031\langnp2057\insrsid2633078\charrsid12468991 }{
\rtlch\fcs1 \ab\af1\afs20 \ltrch\fcs0 \fs20\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid12468991 Serhan, C. N.; Petasis, N. A. }{\rtlch\fcs1 \ab\af1\afs20 \ltrch\fcs0 \i\fs20\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid12468991
Chem Rev}{\rtlch\fcs1 \ab\af1\afs20 \ltrch\fcs0 \fs20\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid12468991 }{\rtlch\fcs1 \ab\af1\afs20 \ltrch\fcs0 \b\fs20\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid12468991 2011}{\rtlch\fcs1
\ab\af1\afs20 \ltrch\fcs0 \fs20\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid12468991 , }{\rtlch\fcs1 \ab\af1\afs20 \ltrch\fcs0 \i\fs20\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid12468991 111}{\rtlch\fcs1 \ab\af1\afs20 \ltrch\fcs0
\fs20\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid12468991 , 5922.
\par }\pard \ltrpar\qj \fi-567\li567\ri0\widctlpar\tx9356\wrapdefault\faauto\adjustright\rin0\lin567\itap0\pararsid12468991 {\rtlch\fcs1 \ab\af1\afs20 \ltrch\fcs0 \fs20\lang2057\langfe1031\langnp2057\insrsid2633078\charrsid12468991 (2) }{\rtlch\fcs1
\ab\af1\afs20 \ltrch\fcs0 \fs20\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid12468991 Chen, P.; Fenet, B.; Michaud, S.; Tomczyk, N.; Vericel, E.; Lagarde, M.; Guichardant, M. }{\rtlch\fcs1 \ab\af1\afs20 \ltrch\fcs0
\i\fs20\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid12468991 FEBS Lett}{\rtlch\fcs1 \ab\af1\afs20 \ltrch\fcs0 \fs20\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid12468991 }{\rtlch\fcs1 \ab\af1\afs20 \ltrch\fcs0
\b\fs20\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid12468991 2009}{\rtlch\fcs1 \ab\af1\afs20 \ltrch\fcs0 \fs20\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid12468991 , }{\rtlch\fcs1 \ab\af1\afs20 \ltrch\fcs0
\i\fs20\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid12468991 583}{\rtlch\fcs1 \ab\af1\afs20 \ltrch\fcs0 \fs20\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid12468991 , 3478.
\par }\pard \ltrpar\qj \fi-142\li142\ri0\widctlpar\wrapdefault\faauto\adjustright\rin0\lin142\itap0\pararsid12468991 {\rtlch\fcs1 \ab\af1\afs20 \ltrch\fcs0 \fs20\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid12468991 (3) }{\rtlch\fcs1 \ab\af1\afs20
\ltrch\fcs0 \fs20\lang2057\langfe1031\langnp2057\insrsid2633078\charrsid12468991 }{\rtlch\fcs1 \ab\af1\afs20 \ltrch\fcs0 \fs20\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid12468991 Butovich, I. A. }{\rtlch\fcs1 \ab\af1\afs20 \ltrch\fcs0
\i\fs20\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid12468991 J Lipid Res}{\rtlch\fcs1 \ab\af1\afs20 \ltrch\fcs0 \fs20\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid12468991 }{\rtlch\fcs1 \ab\af1\afs20 \ltrch\fcs0
\b\fs20\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid12468991 2006}{\rtlch\fcs1 \ab\af1\afs20 \ltrch\fcs0 \fs20\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid12468991 , }{\rtlch\fcs1 \ab\af1\afs20 \ltrch\fcs0
\i\fs20\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid12468991 47}{\rtlch\fcs1 \ab\af1\afs20 \ltrch\fcs0 \fs20\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid12468991 , 854.}{\rtlch\fcs1 \ab\af1\afs20 \ltrch\fcs0
\fs20\lang2057\langfe1031\langnp2057\insrsid2766518\charrsid12468991
\par }\pard \ltrpar\qj \li0\ri0\widctlpar\wrapdefault\faauto\adjustright\rin0\lin0\itap0\pararsid12468991 }}\pard\plain \ltrpar\qj \li0\ri0\widctlpar\wrapdefault\faauto\adjustright\rin0\lin0\itap0\pararsid12468991 \rtlch\fcs1 \af1\afs22\alang1025 \ltrch\fcs0
\f1\fs22\lang1031\langfe1031\cgrid\langnp1031\langfenp1031 \sectd \ltrsect\psz9\linex0\headery709\footery709\colsx284\endnhere\sectdefaultcl\sectrsid12468991\sftnbj {\rtlch\fcs1 \ab\af1\afs20 \ltrch\fcs0
\fs20\lang2057\langfe1031\langnp2057\insrsid9721414\charrsid12468991
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